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rProTx-I

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Origin:Thrixopelma pruriens (Peruvian green velvet tarantula)1.  

Source description:Recombinant,E.coli.

M.W.:3988    Purity: >98%    Effective concentration: 10-100nM

Sequence:ECRYWLGGCSAGQTCCKHLVCSRRHGWCVWDGTFS.

Modifications: Disulfide bonds between Cys2-Cys16, Cys9-Cys21, and Cys15-Cys28.

Molecular formula: C171H245N53O47S6.

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Sizes:50ug, 100ug, 5 x 50ug, 5 x 100ug lyophilized powder.

Activity:  ProTx-I inhibits voltage-gated Ca2+ (Cav3.1), K+ (Kv2.1), and all Na+ channels tested (Nav1.2, Nav1.5, Nav1.7 and Nav1.8). The toxin shifts the voltage-dependence of channel activation to more positive potentials.

References:

1. Middleton, R.E.  et al. (2002) Biochemistry, 41, 14734

2. Bosmans, F. et al. (2006)  Mol. Pharmacol.,  69, 419

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