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rAa1 (K+ channel blo...

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Origin:Androctonus australis (Sahara scorpion).

Source description:Recombinant,E.coli.

M.W.:3868     Purity: >98%    Effective concentration: 100nM - 1uM.

Sequence:QNETNKKCQGGSCASVCRRVIGVAAGKCINGRCVCYP.

Modifications: Disulfide bonds between Cys8-Cys28, Cys13-Cys33, and Cys17-Cys35.

Molecular formula: C156H266N54O49S6.

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Sizes:50ug, 100ug, 5 x 50ug, 5 x 100ug lyophilized powder.

Activity:Aa1 is blocker of A-type voltage-gated transient K+ channels of cerebellar granular cells1.2.

References:

1. Pisciotta, M. et al. (1998) Biochem. Biophys. Res. Comm. 242, 287.

2. Pisciotta, M. et al. (1998) Eur. Biophys. J. 27, 69.

3. Pisciotta, M. et al. (2000) Biochim. Biophys. Acta. 1468, 203.

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